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There is actually a reasonable amount of literature on kratom, so it is possible a pharmaceutical product will be derived from it.

Probably the biggest issue with most (at present, all?) pharmaceutical opioids is the side effect of respiratory depression - this kills a lot of people. Because kratom's active alkaloids don't recruit β-arrestin interactions, side effects like respiratory depression, constipation and tolerance are absent or greatly reduced, which should make mitragynine and 7-OH-mitragynine perfect candidates for a new, safe opioid drug[1].

But patents are probably a huge barrier to this ever happening - you can't patent a plant. No new, patentable extraction methods seem to be required, and a patentable, stronger synthetic or semi-synthetic analogue may not exist[2].

[1] http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3926195/

[2] http://pubs.acs.org/doi/abs/10.1021/jacs.6b00360?journalCode...



Thank you, @GordonS! I will go read up about β-arrestin.

If it is scheduled, does that increase the chance of a safe(r) opioid replacement being developed?

And can you kindly point me to some text books/journals or introductory chemistry in order to understand these interactions at a fundamental level?


Here are a few DOIs to look up on sci-hub:

- 10.1093/bja/aer29

- 10.1007/978-3-642-41199-1_22

- 10.1213/01.ANE.0000160588.32007.AD

- 10.1124/mol.106.028258

- 10.1124/jpet.105.087254

- 10.1523/JNEUROSCI.5999-10.2011

I should add that I'm not a chemist, I just have a keen, self-vested interest in analgesic substances.


Actually, you _can_ patent a plant. It's called a plant patent.

35 USC 161 specifically governs plants.


I'm going to guess this is for patenting strains that are bred or genetically modified? E.g. to provide better disease resistance or higher quantities of substances?

I had meant the 'original', 'natural' plant, but a fair point.




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